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9

抑制剂 & 化合物

2

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Cat. No. Product Name Target Signaling Pathways
T0909L Nalidixic acid sodium salt

萘啶酮酸,萘啶酮酸钠,Baktogram,Sodium nalidixate

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Nalidixic acid sodium salt (Baktogram) 是一种喹诺酮类抗生素,对革兰氏阳性和革兰氏阴性细菌均有效。它在较低浓度下有抑菌作用,在较高浓度下有杀菌作用。它抑制 DNA 促旋酶和拓扑异构酶IV 的亚基,并可逆地阻止易感细菌中的 DNA 复制。
T38359 Dup-721

Antibacterial Microbiology/Virology
DuP-721 是广谱的口服有效的抗菌剂,可以抑制多种临床敏感和耐药细菌,特别是结核杆菌M. tuberculosis。
T1001 Dicloxacillin Sodium hydrate

Dicloxacillin sodium salt monohydrate,双氯西林钠,Dicloxacillin sodium monohydrate

Antibacterial; Antibiotic Microbiology/Virology
Dicloxacillin Sodium hydrate 是一种青霉素类窄谱β内酰胺抗生素,可研究革兰氏阳性菌感染。
T124492 Imipenem

N-Formimidoyl thienamycin,MK0787

Antifungal Microbiology/Virology
Imipenem (MK0787) 是一种噻吩霉素衍生物,属于抗生素类,具有抗菌活性,对革兰氏阳性和革兰氏阴性菌具有部分的抑制作用。Imipenem 可用于研究碳青霉烯类非易感性感染和铜绿假单胞菌生物膜感染。
T33359 Meticillin

Staphcillin,Methicillin,Dimethoxyphenyl Penicillin,Metin

Methicillin is a narrow-spectrum beta-lactam antibiotic of the penicillin-like family, used to treat infections caused by susceptible gram-positive bacteria, in particular penicillase-producing organisms such as Staphylococcus aureus.
T73911 Antibacterial agent 12

Antibacterial agent 12 是一种联芳基恶唑烷酮类似物,是一种针对抗生素敏感和耐药革兰氏阳性菌的抗菌剂。
T37881 Oritavancin(LY-333328)

Oritavancin is a novel semisynthetic glycopeptide antibiotics. On August 6, 2014, the FDA approved oritavancin for treatment of skin infections. Oritavancin possesses potent and rapid bactericidal activity in vitro against a broad spectrum of both resistant and susceptible Gram-positive bacteria, including Staphylococcus aureus, MRSA, enterococci, and streptococci.
T32669 Leucomycin a5

Leukomycin A5,Turimycin H4

Leucomycin a5 is a metabolite from the leucomycin complex, which was originally isolated from S. kitasatoensis. It is active against a variety of Gram-positive and Gram-negative bacteria (MICs = 0.04-0.8 µg/ml) but not against K. pneumoniae, S. typhimuriu
T74803 Levonadifloxacin

Levonadifloxacin ((S)-(-)-Nadifloxacin; WCK 771),作为一种宽谱抗葡萄球菌药物,对甲氧西林敏感金黄色葡萄球菌(MSSA)及对甲氧西林耐药金黄色葡萄球菌(MRSA)显示出显著的抗菌活性,并能有效减少THP-1单核细胞对MRSA和MSSA菌株的吞噬。

化合物

Nalidixic acid sodium salt
Cat.No: T0909L
Synonym: 萘啶酮酸,萘啶酮酸钠,Baktogram,Sodium nalidixate
Target: Topoisomerase, Antibacterial, Antibiotic
Dup-721
Cat.No: T38359
Synonym:
Target: Antibacterial
Dicloxacillin Sodium hydrate
Cat.No: T1001
Synonym: Dicloxacillin sodium salt monohydrate,双氯西林钠,Dicloxacillin sodium monohydrate
Target: Antibacterial, Antibiotic
Imipenem
Cat.No: T124492
Synonym: N-Formimidoyl thienamycin,MK0787
Target: Antifungal
Meticillin
Cat.No: T33359
Synonym: Staphcillin,Methicillin,Dimethoxyphenyl Penicillin,Metin
Target:
Antibacterial agent 12
Cat.No: T73911
Synonym:
Target:
Oritavancin(LY-333328)
Cat.No: T37881
Synonym:
Target:
Leucomycin a5
Cat.No: T32669
Synonym: Leukomycin A5,Turimycin H4
Target:
Levonadifloxacin
Cat.No: T74803
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T0909 Nalidixic acid

萘啶酸,NSC-82174

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Nalidixic acid (NSC-82174) 是一种喹诺酮类抗生素,对革兰氏阳性和革兰氏阴性细菌有效。它在较低浓度下有抑菌作用,而在较高浓度下有杀菌作用。它抑制 DNA 促旋酶和拓扑异构酶 IV 的亚基,并可逆地阻止易感细菌中的 DNA 复制。
T35751 Violacein

Violacein is a bacterial metabolite originally isolated from C. violaceum that has antibacterial and antiprotozoal activities.[1] [2] It is produced by C. violaceum as a purple pigment in response to N-hexanoyl homoserine lactone , a property that has been modified to create a strain of C. violaceum used in detecting quorum-sensing molecules.[3] Violacein is active against Gram-positive bacteria, including B. subtilis and S. aureus (MICs = 0.8 and 1.6 &#181M, respectively). It is also active aga...

天然产物

Nalidixic acid
Cat.No: T0909
Synonym: 萘啶酸,NSC-82174
Target: Topoisomerase, Antibacterial, Antibiotic
Violacein
Cat.No: T35751
Synonym:
Target:
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